From: 99mTc-HYNIC-(tricine/EDDA)-FROP peptide for MCF-7 breast tumor targeting and imaging
99mTc-HYNIC-FROP | |||
---|---|---|---|
%ID/g | |||
15 min | 30 min | Block-15 min | |
Tissue | |||
Blood | 0.48 ± 0.09 | 0.35 ± 0.10 | 0.69 ± 0.16 |
Heart | 0.49 ± 0.08 | 0.26 ± 0.11 | 0.45 ± 0.03 |
Lung | 0.45 ± 0.08 | 0.41 ± 0.26 | 0.60 ± 0.04 |
S.Ta | 0.25 ± 0.03 | 0.32 ± 0.22 | 0.25 ± 0.01 |
Liver | 0.20 ± 0.02 | 0.14 ± 0.00 | 0.26 ± 0.04 |
Spleen | 0.15 ± 0.01 | 0.28 ± 0.11 | 0.23 ± 0.07 |
Kidney | 2.22 ± 0.16 | 1.73 ± 0.15 | 2.97 ± 0.23 |
Stomach | 0.21 ± 0.01 | 0.33 ± 0.12 | 0.26 ± 0.01 |
Muscle | 0.08 ± 0.01 | 0.21 ± 0.16 | 0.15 ± 0.01 |
Bone | 0.18 ± 0.02 | 0.24 ± 0.12 | 0.22 ± 00 |
Intestine | 0.34 ± 0.09 | 0.79 ± 0.25 | 0.64 ± 0.09 |
Tumor | 0.25 ± 0.02 | 0.38 ± 0.21 | 0.09 ± 0.02 |
Tumor/Tissue | |||
Muscle | 3.03 ± 0.12 | 1.94 ± 0.46 | 0.60 ± 0.12 |
Blood | 0.53 ± 0.15 | 1.09 ± 0.47 | 0.14 ± 0.06 |
Spleen | 1.61 ± 0.22 | 1.56 ± 1.04 | 0.42 ± 0.14 |
Bone | 1.36 ± 0.28 | 1.57 ± 0.48 | 0.40 ± 0.09 |
Liver | 1.24 ± 0.28 | 2.62 ± 1.38 | 0.36 ± 0.13 |