Inhibitors | IC50 average µg/mL | Range (µg/mL) | SD | Potency vs | |
---|---|---|---|---|---|
Porcine Gastric Mucin = 1 | Chondroitin sulfate = 1 | ||||
Dextrans | Â | Â | Â | Â | Â |
 Dextran sulfate-500 kDa | 0.018 | 0.001–0.066 | 0.021 | 1892.000 | 25,909.536 |
 Dextran sulfate 6–11 kDa | 0.194 | 0.046–0.962 | 0.242 | 171.926 | 2354.401 |
 Dextran 450 kDa | NSI | NSI | NSI | NSI | NSI |
 Dextran 9–10 kDa | NSI | NSI | NSI | NSI | NSI |
Fucoidans and mucin | Â | Â | Â | Â | Â |
 Macrosystis pyrifera | 0.277 | 0.113–0.423 | 0.096 | 120.529 | 1650.556 |
 Undaria pinnatifada | 0.430 | 0.183–9.77 | 0.252 | 77.600 | 1062.674 |
 Fucus vesiculosus crude | 0.491 | 0.111–1.54 | 0.318 | 67.947 | 930.479 |
 Ascophyllum nodusum nutri. 0.5% | 0.736 | 0.405–1.29 | 0.335 | 45.352 | 621.067 |
 A. nodusum + L. digitata (PS-II) | 0.764 | 0.113–0.423 | 0.096 | 43.649 | 597.734 |
 Fucus vesiculosus 95% | 1.008 | 0.21–2.797 | 0.760 | 33.107 | 453.375 |
 κ-carrageenan | 1.101 | 0.667–1.883 | 0.390 | 30.301 | 414.948 |
 Fucus serratus | 1.520 | 0.203–3.099 | 0.796 | 21.954 | 300.648 |
 F. vesiculosus HCl 10′ 30 kDa | 1.690 | 0.1–2.828 | 0.685 | 19.749 | 270.443 |
 F. vesiculosus Aus. 30 kDa | 2.547 | 0.656–7.066 | 0.501 | 13.100 | 179.396 |
 F. vesiculosus—nutri. 0.5% | 2.924 | 0.331–9.67 | 3.908 | 11.411 | 156.262 |
 F. vesiculosus HCl 10' mix | 5.468 | 3.215–5.215 | 1.520 | 6.102 | 83.568 |
 Laminaria digitata | 5.593 | 0.227–21.0 | 5.983 | 5.966 | 81.698 |
 L. japonica | 21.103 | 9.67–44.447 | 9.806 | 1.581 | 21.654 |
 Porcine Gastric Mucin Type III | 33.368 | 10.156–75.117 | 15.115 | 1.000 | 13.694 |
 A. nodusum | 39.886 | 7.51–71.197 | 18.179 | 0.837 | 11.456 |
 F. vesiculosus HCl 60′ 30 kDa | 59.022 | 13.92–113.723 | 34.505 | 0.565 | 7.742 |
 F. vesiculosus HCl 60' mix | 68.958 | 48.184–86.822 | 23.351 | 0.484 | 6.627 |
 l-Fucose, d-Fucose, Fuc-BSA, methyl-b-Fuc, methyl-a-Fuc | NSI | NSI | NSI | NSI | NSI |
Glycosaminoglycans | Â | Â | Â | Â | Â |
 Chondroitin sulfate-Sigma | 456.950 | 369.911–674.852 | 87.803 | 0.073 | 1.000 |
 Heparin, heparan sulfate, keratan sulfate | NSI | NSI | NSI | NSI | NSI |
Alginates | Â | Â | Â | Â | Â |
 A. nodusum alginate | 3.587 | 1.243–7.81 | 2.210 | 9.301 | 127.375 |
 Alginic acid | 4.931 | 0.975–13.49 | 5.053 | 6.767 | 92.665 |
 L. japonica alginate | 34.228 | 15.439–55.329 | 11.284 | 0.975 | 13.350 |
 Azotobacter spp. alginate | NSI | NSI | NSI | NSI | NSI |
Others | Â | Â | Â | Â | Â |
 Lotus lectin (LTL) | 17.564 | 13.943–27.717 | 8.408 | 3.968 | 26.015 |
 Sambucus Nigra lectin (SNA) | 52.924 | 42.695–631.54 | 14,466 | 2.306 | 8.633 |
 Concanavalin A lectin (ConA) | 140.943 | 79.19–237.597 | 84.774 | 0.393 | 3.242 |
 Blood Group Lewis-B | 471.548 | 7.919–23.760 | 60.393 | 0.552 | 0.969 |